What is the catalog number for TM-1?

The catalog number for TM-1 is T63012.

What sizes are available for TM-1?

TM-1 is available in the following size(s): 100 mg, 25 mg, 50 mg.

How many pack sizes does TM-1 come in?

TM-1 is available in 3 different pack sizes.

TM-1 is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures TM-1?

TM-1 is manufactured by Molfinity.

What is the estimated delivery time for TM-1?

Estimated delivery time for TM-1 is approximately 10 business day(s), depending on your location.

TM-1

Product Specifications

CAS Number

921099-13-0

Target

Others, Dehydrogenase

Related Pathways

Metabolism, Others

Bioactivity

TM-1 is a potent pyruvate dehydrogenase kinase (PDHK) inhibitor that inhibits the activity of PDHK1 (IC50: 2.97 μM) and PDHK2 (IC50: 5.2 μM) . TM-1 blocks pyruvate dehydrogenase complex (PDHC) phosphorylation and inhibits cancer cell proliferation.