CCG-271423
Product Specifications
CAS Number
2750413-88-6
Target
GRK|||Others
Related Pathways
Others|||GPCR/G Protein
Bioactivity
CCG-271423 is a potent and selective inhibitor of GRK5, demonstrating activity against GRK5 (IC50: 0.0021 ?M) and GRK2 (IC50: 44 ?M) ; it reduces Ca2+ transients and inhibits cardiomyocyte contractility.
Smiles
C(=C\1/C=2C(NC1=O)=CC=C(C(N[C@H](C)C3=CC=CC=C3)=O)C2)\C4=C(C)C(C(NCC#C)=O)=C(C)N4
Molecular Formula
C28H26N4O3
Molecular Weight
466.53
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
Curated Selection
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