CCG-271423
Product Specifications
CAS Number
2750413-88-6
Target
GRK|||Others
Related Pathways
Others|||GPCR/G Protein
Bioactivity
CCG-271423 is a potent and selective inhibitor of GRK5, demonstrating activity against GRK5 (IC50: 0.0021 ?M) and GRK2 (IC50: 44 ?M) ; it reduces Ca2+ transients and inhibits cardiomyocyte contractility.
Smiles
C(=C\1/C=2C(NC1=O)=CC=C(C(N[C@H](C)C3=CC=CC=C3)=O)C2)\C4=C(C)C(C(NCC#C)=O)=C(C)N4
Molecular Formula
C28H26N4O3
Molecular Weight
466.53
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
Curated Selection
Explore Other Products
Discover premium biology products from our extensive collection of 20M+ items
127591-PE 100 µL
GSTA3 (Glutathione S-transferase A3, GST Class-alpha Member 3, Glutathione S-transferase A3-3, MGC22232) (PE)
Ask
View Details 
GTR15300684 1 Vial
Lentiviral mouse Znhit1 shRNA (UAS) - Lentiviral mouse Znhit1 shRNA (UAS, GFP) (100)
Ask
View Details 