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SHR2415

Product Specifications

Target

Others|||ERK

Related Pathways

Others|||MAPK

Bioactivity

SHR2415 is a selective, potent, orally active inhibitor of ERK1/2. SHR2415 inhibits ERK1 (IC50: 2.8 nM) and ERK2 (IC50: 5.9 nM) . SHR2415 exhibits high potency in Colo205 cells (IC50: 44.6 nM) . SHR2415 can be used in cancer research.

Molecular Formula

C23H22ClN7O2

Molecular Weight

463.92

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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