GPR84 antagonist 3
Product Specifications
CAS Number
2815263-05-7
Target
Others, GPCR
Related Pathways
Others, Endocrinology/Hormones, GPCR/G Protein
Bioactivity
GPR84 Antagonist 3 (compound 42), a potent inhibitor of the G-protein-coupled receptor 84 (GPR84), exhibits a pIC50 value of 8.28, indicating strong antagonistic activity by inhibiting GTPγS. Additionally, it possesses a favorable pharmacokinetic profile, suitable for further research and development [1].
Smiles
C(C=1N=C(C(=NN1)C2=CC=C(CN3CCOCC3)C=C2)C4=CC=CC=C4)C=5C=6C(NC5)=CC=CC6
Molecular Formula
C29H27N5O
Molecular Weight
461.56
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
E-OSEL-R0008-01 24 Tests
QuicKey Pro Rat IL-1R2 (Interleukin 1 Receptor Type II) ELISA Kit
Sign In for Pricing
View Details E-OSEL-R0008-02 48 Tests
QuicKey Pro Rat IL-1R2 (Interleukin 1 Receptor Type II) ELISA Kit
Sign In for Pricing
View Details