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RET-IN-7

Product Specifications

CAS Number

2763386-05-4

Target

C-RET, Others

Related Pathways

Tyrosine Kinase/Adaptors, Others, Apoptosis

Bioactivity

RET-IN-7 exhibits strong inhibitory effects against RET kinase in vitro and shows significant efficacy in treating RET-driven tumor xenografts in mice through multiple-day dosing.

Smiles

N(C(OC)=O)C12CCC(CC1)(CC2)N3C=4C(C(=C3)C5=C(F)C=C(Cl)C(N)=C5)=C(N)N=CN4

Molecular Formula

C22H24ClFN6O2

Molecular Weight

458.92

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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