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PDGFR-IN-1

Product Specifications

CAS Number

2644673-07-2

Target

PDGFR, Apoptosis

Related Pathways

Tyrosine Kinase/Adaptors, Angiogenesis, Apoptosis

Purity

0.9949

Bioactivity

PDGFR-IN-1 is an orally active, highly efficient platelet-derived growth factor receptor (PDGFR) inhibitor with potent antitumor activity. It inhibits PDGFRα and PDGFRβ and can be used in solid tumor research.

Smiles

N1=CC=2C=CC(=CC2N1)NC3=NC(=NC=C3C)NC4=CC=C(C(OC)=C4)N5CCN(CC)CC5

Molecular Formula

C25H30N8O

Molecular Weight

458.56

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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