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FLT3/TrKA-IN-1

Product Specifications

Target

Apoptosis|||FLT|||Others|||Trk receptor

Related Pathways

Tyrosine Kinase/Adaptors|||Others|||Angiogenesis|||Apoptosis

Bioactivity

FLT3/TrKA-IN-1 is a potent dual kinase inhibitor that targets FLT3 (IC50: 43.8 nM), FLT3-ITD (IC50: 97.2 nM), FLT3-TKD (IC50: 92.5 nM), and TrKA (IC50: 23.6 nM) . FLT3/TrKA-IN-1 shows potential for acute myeloid leukaemia (AML) studies.

Molecular Formula

C28H30N4O2

Molecular Weight

454.56

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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