GPR81 agonist 1
Product Specifications
CAS Number
1620992-67-7
Target
GPCR, HCAR
Related Pathways
GPCR/G Protein, Endocrinology/Hormones
Purity
0.9968
Bioactivity
GPR81 agonist 1 is a potent and selective GPR81 agonist with high affinity for human and mouse GPR81, inhibiting lipolysis of differentiated 3T3-L1 adipocytes, improving insulin sensitivity and glycaemic control in mouse models of insulin resistance and diabetes, and can be used in the study of diabetes and obesity.
Smiles
C[C@H]1CC[C@@H](CC1)C(=O)Nc1nc(c(CC(=O)N2CCN(C)CC2)s1)-c1cccs1
Molecular Formula
C22H30N4O2S2
Molecular Weight
446.63
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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