GRK5-IN-3

Product Specifications

CAS Number

2410793-22-3

Target

Others, GRK

Related Pathways

Others, GPCR/G Protein

Bioactivity

GRK5-IN-3 is a covalent inhibitor of G protein-coupled receptor kinase 5 (GRK5), significantly inhibiting GRK5 with an IC50 of 0.22 μM and GRK6 with an IC50 of 0.41 μM.

Smiles

N(C1=C2C(=NC(NC3=C(OC)C=C(NC(C=C)=O)C=C3)=N1)NC=C2)C4=C(C(N)=O)C=CC=C4

Molecular Formula

C23H21N7O3

Molecular Weight

443.46

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

More Discoveries

Explore Other Products

Browse additional items from our catalog

orb2941480-01 250 mg

1,2:4,6-Bis-O- (1-methylethylidene) -L-sorbofuranose

View Details

orb2941480-02 100 mg

1,2:4,6-Bis-O- (1-methylethylidene) -L-sorbofuranose

View Details

orb2941480-03 50 mg

1,2:4,6-Bis-O- (1-methylethylidene) -L-sorbofuranose

View Details

AMM09299V 100 µL

Leukotriene A4 hydrolase (LTA4H) Mouse Monoclonal Antibody [Clone ID: LBI9G8]

View Details

SI000185A 1 Each

Human ACSBG1 Pre-designed siRNA Set A

View Details

22114034 100 µg

Gm5634 Protein Lysate (Mouse) with C-HA Tag

View Details