GRK5-IN-3

Product Specifications

CAS Number

2410793-22-3

Target

Others|||GRK

Related Pathways

Others|||GPCR/G Protein

Bioactivity

GRK5-IN-3 is a covalent inhibitor of G protein-coupled receptor kinase 5 (GRK5), significantly inhibiting GRK5 with an IC50 of 0.22 ?M and GRK6 with an IC50 of 0.41 ?M.

Smiles

N(C1=C2C(=NC(NC3=C(OC)C=C(NC(C=C)=O)C=C3)=N1)NC=C2)C4=C(C(N)=O)C=CC=C4

Molecular Formula

C23H21N7O3

Molecular Weight

443.46

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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