GRK5-IN-3
Product Specifications
CAS Number
2410793-22-3
Target
Others|||GRK
Related Pathways
Others|||GPCR/G Protein
Bioactivity
GRK5-IN-3 is a covalent inhibitor of G protein-coupled receptor kinase 5 (GRK5), significantly inhibiting GRK5 with an IC50 of 0.22 ?M and GRK6 with an IC50 of 0.41 ?M.
Smiles
N(C1=C2C(=NC(NC3=C(OC)C=C(NC(C=C)=O)C=C3)=N1)NC=C2)C4=C(C(N)=O)C=CC=C4
Molecular Formula
C23H21N7O3
Molecular Weight
443.46
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
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