PPARγ phosphorylation inhibitor 1
Product Specifications
CAS Number
2882975-84-8
Target
PPAR
Related Pathways
Metabolism, DNA Damage/DNA Repair
Purity
0.9986
Bioactivity
PPARγ phosphorylation inhibitor 1 (Compound 10) is an effective PPARγ agonist (IC50=24 nM) that inhibits CDK5-mediated PPARγ Ser273 phosphorylation (IC50=160 nM) and exhibits antidiabetic activity.
Smiles
O=C(O)C1=NN(C(=O)C=2C=C(OC=3C=CC=CC3)C=CC12)CC4=CC=C(Cl)C(Cl)=C4
Molecular Formula
C22H14Cl2N2O4
Molecular Weight
441.26
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
MBS6192572-01 0.1 mL
SREK1 (Splicing Regulatory Glutamine/lysine-rich Protein 1, Serine/arginine-rich-splicing Regulatory Protein 86, SRrp86, Splicing Factor, Arginine/serine-rich 12, SFRS12, Splicing Regulatory Protein 508, SRrp508) (MaxLight 405)
Sign In for Pricing
View Details MBS6192572-02 5x 0.1 mL
SREK1 (Splicing Regulatory Glutamine/lysine-rich Protein 1, Serine/arginine-rich-splicing Regulatory Protein 86, SRrp86, Splicing Factor, Arginine/serine-rich 12, SFRS12, Splicing Regulatory Protein 508, SRrp508) (MaxLight 405)
Sign In for Pricing
View Details 