A2AAR/HDAC-IN-1

2767560-51-8

Adenosine Receptor, Others, HDAC

Chromatin/Epigenetic, Others, Neuroscience, DNA Damage/DNA Repair, GPCR/G Protein

A2AAR/HDAC-IN-1 (compound 14c) is an orally active, balanced dual inhibitor of A2AAR (Ki: 163.5 nM) and HDAC1 (IC50: 145.3 nM) .

C(CC1=CC=C(C(NC2=C(N)C=CC=C2)=O)C=C1)N3C=4C(=C(N=C(N)N4)C5=CC=CO5)C=N3

C24H21N7O2

439.47

Ice Packs

-20°C