CB1/2 agonist 1
Product Specifications
Target
Others, Cannabinoid Receptor
Related Pathways
Others, GPCR/G Protein
Bioactivity
CB1/2 agonist 1 is a potent CB1/2 agonist that crosses the blood-brain barrier, acting on CB1R (EC50: 56.15 nM) and CB2R (EC50: 11.63 nM) . It reduces glutamate release and LPS-induced microglia activation, exhibiting anti-inflammatory and analgesic activities, with potential for multiple sclerosis studies.
Molecular Formula
C21H24BrFN2O2
Molecular Weight
435.33
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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