GABAA receptor agent 2 TFA
Product Specifications
CAS Number
1781880-44-1
Target
GABA Receptor, Others
Related Pathways
Neuroscience, Others, Membrane transporter/Ion channel
Bioactivity
GABAA receptor agent 2 TFA is a potent, high-affinity GABAA receptor antagonist with an IC50 of 24 nM [human α1β2γ2GABAA-expressing tsA201 cells] and a Ki of 28 nM [rat GABAA receptor]. GABAA receptor agent 2 TFA has no effect on four human GABA transport proteins [hGAT-1, hBGT-1, hGAT-2, and hGAT-3].
Smiles
O=C(O)C(F)(F)F.ON1N=CC(=C1C=2C=CC=C(C2)C=3C=CC=CC3)C4CCNCC4
Molecular Formula
C22H22F3N3O3
Molecular Weight
433.42
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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