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PI3Kδ-IN-11

Product Specifications

CAS Number

2413257-51-7

Target

Apoptosis, Akt, Others, PI3K

Related Pathways

Others, PI3K/Akt/mTOR signaling, Apoptosis, Cytoskeletal Signaling

Bioactivity

PI3Kδ-IN-11 is a potent and selective PI3Kδ inhibitor (IC50: 27.5 nM) that dose-dependently blocks PI3K/Akt pathway activity. PI3Kδ-IN-11 can be used in B- or T-cell-associated malignancy studies.

Smiles

N(C=1C2=C(C=CC(=C2)C3=CC4=C(N=C3)C=CC=C4)N=CN1)C5=CC(NC(C=C)=O)=C(C)C=C5

Molecular Formula

C27H21N5O

Molecular Weight

431.49

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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