PI3Kδ-IN-11
Product Specifications
CAS Number
2413257-51-7
Target
Apoptosis, Akt, Others, PI3K
Related Pathways
Others, PI3K/Akt/mTOR signaling, Apoptosis, Cytoskeletal Signaling
Bioactivity
PI3Kδ-IN-11 is a potent and selective PI3Kδ inhibitor (IC50: 27.5 nM) that dose-dependently blocks PI3K/Akt pathway activity. PI3Kδ-IN-11 can be used in B- or T-cell-associated malignancy studies.
Smiles
N(C=1C2=C(C=CC(=C2)C3=CC4=C(N=C3)C=CC=C4)N=CN1)C5=CC(NC(C=C)=O)=C(C)C=C5
Molecular Formula
C27H21N5O
Molecular Weight
431.49
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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