Cabotegravir sodium
Product Specifications
CAS Number
1051375-13-3
Target
Others, HIV Protease, OAT
Related Pathways
Membrane transporter/Ion channel, Others, Microbiology/Virology, Proteases/Proteasome
Purity
0.9963
Bioactivity
Cabotegravir sodium (GSK-1265744) is an orally active, membrane-permeable HIV integrase inhibitor (IC50 = 2.5 μM) and also an OAT1/OAT3 inhibitor (IC50 = 0.81/0.41 μM) . It inhibits HIV replication and may be used in AIDS research.
Smiles
[Na+].C[C@H]1CO[C@@H]2Cn3cc(C(=O)NCc4ccc(F)cc4F)c(=O)c([O-])c3C(=O)N12
Molecular Formula
C19H16F2N3NaO5
Molecular Weight
427.34
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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