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TLR7/8 antagonist 1

Product Specifications

Target

TLR, Others

Related Pathways

Immunology/Inflammation, Others

Bioactivity

TLR7/8 Antagonist 1 (Compound 16c), an imidazoquinoline derivative, is a potent TLR7/8 agonist with IC50 values of 3.91 and 2.19 μM for TLR7 and TLR8, respectively. rel-O-2050 (TLR-2050) is a key target for drug development in infectious diseases, cancer, and autoimmune diseases.

Molecular Formula

C24H27N5O2

Molecular Weight

417.5

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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