LP-922761 hydrate
Product Specifications
Target
Others, AAK1 (AP2 associated kinase 1)
Related Pathways
Others, Neuroscience
Bioactivity
LP-922761 hydrate is a selective, potent, orally active AAK1 inhibitor with IC50 values of 4.8 nM and 7.6 nM in enzyme and cellular assays, respectively. LP-922761 hydrate inhibits BMP-2 inducible protein kinase (BIKE) (IC50: 24 nM) . 922761 hydrate has no significant effect on cellular GAK, opioids, adrenergic α2 or GABAa receptors.
Molecular Formula
C21H28N6O4
Molecular Weight
414.98
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
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