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CDK8-IN-6

Product Specifications

CAS Number

2415156-27-1

Target

Others, CDK

Related Pathways

Cell Cycle/Checkpoint, Others

Bioactivity

CDK8-IN-6 (compound 9) is a potent inhibitor of cyclin-dependent kinase 8 (CDK8) with a Kd of 13 nM, demonstrating significant research potential in AML cancers.

Smiles

C[C@@]12[C@]([C@]3([C@](CC1)([C@]4(C)[C@@](CC3)(C[C@H](N(C)C)CC4)[H])[H])[H])(CC=C2C=5C=C(Cl)C=NC5)[H]

Molecular Formula

C26H37ClN2

Molecular Weight

413.04

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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