Topo I/COX-2-IN-1
Product Specifications
Target
Others, Apoptosis, Prostaglandin Receptor, Topoisomerase
Related Pathways
Apoptosis, GPCR/G Protein, Others, DNA Damage/DNA Repair, Immunology/Inflammation
Bioactivity
Topo I/COX-2-IN-1 (1H-30) is a potent Topo I/COX-2 inhibitor with IC50 values of 0.24 μM for COX-2 and 4.42 μM for Topo I. It induces apoptosis and inhibits cancer cell migration, demonstrating anti-cancer activity.
Molecular Formula
C21H18ClFN2O3
Molecular Weight
400.83
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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