Adenosine receptor inhibitor 1
Product Specifications
CAS Number
2550400-52-5
Target
Adenosine Receptor, Others
Related Pathways
GPCR/G Protein, Others, Neuroscience
Bioactivity
Adenosine receptor inhibitor 1 is a highly potent and selective antagonist of adenosine receptor (AR), exhibiting exceptional affinity for A1 AR, A2A AR, A2B AR, and A3 AR, with respective Ki values of >1000, 68.5, >1000, >1000 nM. This compound demonstrates notable antinociceptive, anti-inflammatory, and peripheral analgesic properties, holding great promise for investigating cancer and neurodegenerative diseases [1].
Smiles
CN1C2=C(N(C)C(NCC3=C(F)C(OC)=CC=C3Cl)=N2)C(=O)N(CC)C1=O
Molecular Formula
C17H19ClFN5O3
Molecular Weight
395.82
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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