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PARP-1-IN-1

Product Specifications

Target

Others|||PARP

Related Pathways

DNA Damage/DNA Repair|||Others|||Chromatin/Epigenetic

Bioactivity

PARP-1-IN-1 is a highly selective and orally active inhibitor of the enzyme PARP-1 with an IC50 of 0.96 nM, exhibiting excellent tolerance and significant activity in a single dose in the MDA-MB-436 xenotransplantation model [1].

Molecular Formula

C23H25FN4O

Molecular Weight

392.47

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Product Datasheet

https://www.targetmol.com/attachment/DataSheet/0B38E7DA-1825-4DB3-B44B-D05911F9ECC6/T61798

Available Sizes

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