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MtTMPK-IN-1

Product Specifications

Target

DNA/RNA Synthesis|||Others|||Antibacterial

Related Pathways

DNA Damage/DNA Repair|||Cell Cycle/Checkpoint|||Others|||Microbiology/Virology

Bioactivity

MtTMPK-IN-1 (compound 3) is a highly effective inhibitor of Mycobacterium tuberculosis thymidylate kinase (Mt TMPK), with an IC50 value of 2.5 ?M. It shows moderate to weak activity against Mtb H37Rv and low cytotoxicity in human fibroblast cells MRC-5, making it a valuable tool for tuberculosis research [1].

Molecular Formula

C22H24N4O3

Molecular Weight

392.45

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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