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TRPV1 antagonist 3

Product Specifications

Target

Others, TRP/TRPV Channel

Related Pathways

Membrane transporter/Ion channel, Others

Bioactivity

TRPV1 antagonist 3 (Compound 7q) is a highly potent TRPV1 receptor antagonist with an IC50 of 2.66 nM against capsaicin. It exhibits selectivity in its mode of action, is orally bioavailable (60%), and can penetrate the central nervous system [1].

Molecular Formula

C23H25N3OS

Molecular Weight

391.53

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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