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Keap1-Nrf2-IN-4

Product Specifications

Target

Apoptosis|||E1/E2/E3 Enzyme|||Others

Related Pathways

Others|||Ubiquitination|||Apoptosis

Bioactivity

Keap1-Nrf2-IN-4, a powerful neddylation inhibitor, demonstrates significant anti-proliferation activity against MGC-803 cells (IC50 = 2.55 ?M), effectively impeding their migration and inducing apoptosis. Additionally, it effectively inhibits tumor growth while exhibiting minimal toxicity [1].

Molecular Formula

C26H34N2O

Molecular Weight

390.56

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Product Datasheet

https://www.targetmol.com/attachment/DataSheet/2FBC7C15-3A7E-4A9D-A1E2-644E41C993A3/T61773

Available Sizes

Curated Selection

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