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Keap1-Nrf2-IN-4

Product Specifications

Target

Apoptosis, E1/E2/E3 Enzyme, Others

Related Pathways

Others, Ubiquitination, Apoptosis

Bioactivity

Keap1-Nrf2-IN-4, a powerful neddylation inhibitor, demonstrates significant anti-proliferation activity against MGC-803 cells (IC50 = 2.55 μM), effectively impeding their migration and inducing apoptosis. Additionally, it effectively inhibits tumor growth while exhibiting minimal toxicity [1].

Molecular Formula

C26H34N2O

Molecular Weight

390.56

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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