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Trk-IN-8

Product Specifications

Target

Others|||Trk receptor

Related Pathways

Tyrosine Kinase/Adaptors|||Others

Bioactivity

Trk-IN-8, a powerful TRK inhibitor, demonstrates excellent potency against TRKAa, TRKA (G595R), and TRKC (G623R) with IC50 values of 0.42 nM, 0.89 nM, and 1.5 nM, respectively (WO2021115401A1, compound 3) [1].

Molecular Formula

C18H16F2N6O2

Molecular Weight

386.36

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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