What is the catalog number for AAK1-IN-5?

The catalog number for AAK1-IN-5 is T61693.

What sizes are available for AAK1-IN-5?

AAK1-IN-5 is available in the following size(s): 25 mg, 50 mg, 100 mg.

How many pack sizes does AAK1-IN-5 come in?

AAK1-IN-5 is available in 3 different pack sizes.

Is AAK1-IN-5 in stock?

AAK1-IN-5 is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures AAK1-IN-5?

AAK1-IN-5 is manufactured by Molfinity.

What is the estimated delivery time for AAK1-IN-5?

Estimated delivery time for AAK1-IN-5 is approximately 10 business day(s), depending on your location.

AAK1-IN-5

Product Specifications

CAS Number

1815613-44-5

Target

Others, AAK1 (AP2 associated kinase 1)

Related Pathways

Others, Neuroscience

Bioactivity

AAK1-IN-5 is a potent and specific inhibitor of adaptor protein-2-associated kinase 1 (AAK1), characterized by its ability to penetrate the central nervous system and its oral bioavailability. It displays high selectivity, with an AAK1 inhibitory potency (IC 50) of 1.2 nM, a binding affinity (K i) of 0.05 nM, and an inhibitory potency against cellular AAK1 activity (cell IC 50) of 0.5 nM. AAK1-IN-5 holds promise for investigating neuropathic pain in scientific research [1].