ERK5-IN-4
Product Specifications
CAS Number
1888305-17-6
Target
Others, ERK
Related Pathways
Others, MAPK
Bioactivity
ERK5-IN-4 (compound 34b) is a potent and specific inhibitor of extracellular signal-related kinase 5 (ERK5) activity, effectively inhibiting both full-length ERK5 and truncated ERK5 (ERK5 ΔTAD) kinase activity in HEK293 cells with IC50 values of 77 nM and 300 nM, respectively [1].
Smiles
C(=O)(C=1C=C(C(NC=2C=NN(C)C2)=O)NC1)C3=C(F)C(Cl)=CC=C3Cl
Molecular Formula
C16H11Cl2FN4O2
Molecular Weight
381.19
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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