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CXCR2 antagonist 4

Product Specifications

Target

Others, CXCR

Related Pathways

Others, Immunology/Inflammation, GPCR/G Protein, Autophagy

Bioactivity

CXCR2 antagonist 4 (compound 7) is a highly potent inhibitor of CXCR2 with an IC50 of 0.13 μM and effectively inhibits the CXCL8-induced cytosolic calcium increase with an IC50 of 27 μM, demonstrating promising potential for anticancer research [1].

Molecular Formula

C15H14F2N4OS2

Molecular Weight

368.42

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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