MRGPRX4 modulator-1
Product Specifications
CAS Number
2492596-61-7
Target
Others, MRGPR
Related Pathways
GPCR/G Protein, Others
Bioactivity
MRGPRX4 modulator-1 (compound 31-2) is a potent antagonist of the mas-related G-protein receptor X4 (MRGPR X4) with an IC50 < 100 nM against MRGPR4, utilized for investigating MRGPR X4-dependent diseases including itch, pain, and autoimmune disorders [1].
Smiles
C(OC1=C(Cl)C=C(C(F)(F)F)C=C1)C=2N=C(C(O)=O)C=C(CC)C2
Molecular Formula
C16H13ClF3NO3
Molecular Weight
359.73
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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