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EAI001

Product Specifications

CAS Number

892772-75-7

Target

EGFR

Related Pathways

JAK/STAT signaling|||Tyrosine Kinase/Adaptors|||Angiogenesis

Purity

>99.99%

Bioactivity

EAI001 is a potent and selective mutant epidermal growth factor receptor (EGFR) variant inhibitor that inhibits EGFRL858R/T790M with an IC50 value of 24 nM.EAI001 can be used in cancer research.

Smiles

O=C(Nc1nccs1)C(N1Cc2ccccc2C1=O)c1ccccc1

Molecular Formula

C19H15N3O2S

Molecular Weight

349.41

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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