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E7016

Product Specifications

CAS Number

902128-92-1

Target

PARP

Related Pathways

Chromatin/Epigenetic, DNA Damage/DNA Repair

Purity

0.9902

Bioactivity

E7016 (GPI 21016) is an orally available PARP inhibitor that inhibits DNA repair and enhances tumor cell radiosensitivity both in vitro and in vivo.

Smiles

OC1CCN(Cc2ccc3oc4cccc5c4c(n[nH]c5=O)c3c2)CC1

Molecular Formula

C20H19N3O3

Molecular Weight

349.38

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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