E7016
Product Specifications
CAS Number
902128-92-1
Target
PARP
Related Pathways
Chromatin/Epigenetic, DNA Damage/DNA Repair
Purity
0.9902
Bioactivity
E7016 (GPI 21016) is an orally available PARP inhibitor that inhibits DNA repair and enhances tumor cell radiosensitivity both in vitro and in vivo.
Smiles
OC1CCN(Cc2ccc3oc4cccc5c4c(n[nH]c5=O)c3c2)CC1
Molecular Formula
C20H19N3O3
Molecular Weight
349.38
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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