What is the catalog number for GAT564?

The catalog number for GAT564 is T61180.

What sizes are available for GAT564?

GAT564 is available in the following size(s): 25 mg, 50 mg, 100 mg.

How many pack sizes does GAT564 come in?

GAT564 is available in 3 different pack sizes.

GAT564 is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures GAT564?

GAT564 is manufactured by Molfinity.

What is the estimated delivery time for GAT564?

Estimated delivery time for GAT564 is approximately 10 business day(s), depending on your location.

GAT564

Product Specifications

Target

Others, Cannabinoid Receptor

Related Pathways

Others, GPCR/G Protein

Bioactivity

GAT564 (Compound 15d) is a highly effective allosteric modulator of the cannabinoid 1 receptor (CB1R), with EC50 values of 87 nM for cAMP and 320 nM for β-arrestin2. It significantly enhances the binding of orthosteric ligands to hCB1R and exhibits remarkable efficacy as a topical agent, significantly reducing intraocular pressure (IOP) in an ocular normotensive murine model of glaucoma [1].