EMI48
Product Specifications
CAS Number
34564-13-1
Target
EGFR, Others
Related Pathways
Angiogenesis, Tyrosine Kinase/Adaptors, Others, JAK/STAT signaling
Bioactivity
EMI48, a derivative of EMI1, exhibits increased efficacy against mutant EGFR compared to EMI1. It specifically inhibits EGFR triple mutants [1].
Smiles
CCN(CC)c1ccc2cc(-c3nc4cc(C)ccc4o3)c(=O)oc2c1
Molecular Formula
C21H20N2O3
Molecular Weight
348.4
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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