Protein kinase D inhibitor 1
Product Specifications
CAS Number
2489320-03-6
Target
Others, Serine/threonin kinase
Related Pathways
Cell Cycle/Checkpoint, Others, Metabolism
Bioactivity
Protein kinase D inhibitor 1 (compound 17m) is a potent pan-PKD inhibitor with IC50 values between 17 and 35 nM, demonstrating inhibitory activity in the low nanomolar range. By inhibiting protein kinase D, it effectively suppresses PKD-dependent cortactin phosphorylation [1].
Smiles
NC1=C2C(=NN(CC3CCNCC3)C2=NC=N1)C=4C=5C(NC4)=CC=CC5
Molecular Formula
C19H21N7
Molecular Weight
347.42
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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