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EGFR/HER2-IN-8

Product Specifications

Target

Others|||EGFR

Related Pathways

JAK/STAT signaling|||Angiogenesis|||Tyrosine Kinase/Adaptors|||Others

Bioactivity

EGFR/HER2-IN-8 (compound 34) is an inhibitor of EGFR, HER2, and DHFR with IC50 values of 0.45 ?M, 0.244 ?M, and 5.669 ?M, respectively. It demonstrates anticancer activity against several cancer cell lines, exhibiting a high safety profile and selectivity indices, making it useful for cancer research [1].

Molecular Formula

C16H16N4O2S

Molecular Weight

328.39

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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