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RP-6306

Product Specifications

CAS Number

2719793-90-3

Target

Wee1

Related Pathways

Cell Cycle/Checkpoint

Purity

0.9928

Bioactivity

Lunresertib (RP-6306) is a potent, selective, and orally active PKMYT1 inhibitor with an IC50 of 14 nM. Lunresertib (RP-6306) inhibits the growth of CCNE1-amplified tumor cells in several preclinical xenograft models.

Smiles

NC=1N(C=2C(C1C(N)=O)=CC(C)=C(C)N2)C3=C(C)C(O)=CC=C3C

Molecular Formula

C18H20N4O2

Molecular Weight

324.38

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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