Brompheniramine
Product Specifications
CAS Number
86-22-6
Target
AChR, Histamine Receptor, Potassium Channel, Calcium Channel, Others, Sodium Channel
Related Pathways
Metabolism, Others, Membrane transporter/Ion channel, Immunology/Inflammation, GPCR/G Protein, Neuroscience
Bioactivity
Brompheniramine ((±) -Brompheniramine) is a potent, orally active alkylamine class antihistamine and a selective antagonist of the histamine H1 receptor (Kd = 6.06 nM) . It has applications in the research of allergic rhinitis and exhibits anticholinergic, antidepressant, and anesthetic properties. Brompheniramine blocks calcium channels, sodium channels, and hERG channels with IC50 values of 16.12 μM, 21.26 μM, and 0.90 μM, respectively [1] [2] [3] [4].
Smiles
C(CCN(C)C)(C1=CC=C(Br)C=C1)C2=CC=CC=N2
Molecular Formula
C16H19BrN2
Molecular Weight
319.24
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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