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PF-06305591 dihydrate

Product Specifications

Target

Others|||Sodium Channel

Related Pathways

Others|||Membrane transporter/Ion channel

Bioactivity

PF-06305591 dihydrate is a potent and highly selective voltage-gated sodium channel NaV1.8 blocker (IC50 = 15 nM) with excellent preclinical in vitro ADME and safety profiles [1].

Molecular Formula

C15H26N4O3

Molecular Weight

310.39

Shipping Conditions

Cool pack

Storage Temperature

-20°C

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