GSK343
Product Specifications
CAS Number
1346704-33-3
Target
Histone Methyltransferase, Autophagy
Related Pathways
Autophagy, Chromatin/Epigenetic
Purity
0.999
Bioactivity
GSK343, a specific and effective EZH2 inhibitor (IC50=4 nM), exhibits 60 fold specificity activity against EZH1, and >1000 fold specificity activity against other histone methyltransferases.
Smiles
CCCc1cc(C)[nH]c(=O)c1CNC(=O)c1cc(cc2n(ncc12)C(C)C)-c1ccnc(c1)N1CCN(C)CC1
Molecular Formula
C31H39N7O2
Molecular Weight
541.69
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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