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HIF-1α-IN-4

Product Specifications

Target

Others, HIF/HIF Prolyl-Hydroxylase

Related Pathways

Others, Chromatin/Epigenetic, Metabolism

Bioactivity

HIF-1α-IN-4 is an inhibitor of HIF-1α with IC50 of 24 nM in HEK293T cells which has potential antitumor effects. HIF-1α-IN-4 downregulates VEGF and PDK1 mRNA expressions under hypoxia [1].

Molecular Formula

C16H12N2O3

Molecular Weight

280.28

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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