PBRM1-BD2-IN-8
Product Specifications
CAS Number
2819989-75-6
Target
Epigenetic Reader Domain
Related Pathways
Chromatin/Epigenetic
Purity
0.9989
Bioactivity
PBRM1-BD2-IN-8 (compound 34) is a potent PBRM1 Bromodomain inhibitor with PBRM1-BD2 Kd of 4.4 ?M, PBRM1-BD2 IC50 of 0.16 ?M, and PBRM1-BD5 Kd of 25 ?M; PBRM1-BD2-IN-8 shows anti-cancer activity.
Smiles
O=C1C=2C(NC(N1)C3=CC(C)=CC=C3)=CC=CC2Br
Molecular Formula
C15H13BrN2O
Molecular Weight
317.18
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
Curated Selection
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