PBRM1-BD2-IN-2
Product Specifications
CAS Number
2819989-57-4
Target
Epigenetic Reader Domain
Related Pathways
Chromatin/Epigenetic
Purity
>99.99%
Bioactivity
PBRM1-BD2-IN-2, a selective and cell-active inhibitor of the polybromo-1 (PBRM1) bromodomain, exhibits binding affinity and inhibitory activity specifically targeting the PBRM1-BD2 domain, with Kd and IC50 values of 9.3 μM and 1.0 μM, respectively. This compound is utilized in cancer research.
Smiles
O=C1C=2C(NC(N1)C3=C(Cl)C=CC=C3F)=CC=CC2Cl
Molecular Formula
C14H9Cl2FN2O
Molecular Weight
311.14
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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