MSC-4106
Product Specifications
CAS Number
2738542-58-8
Target
YAP
Related Pathways
Stem Cells
Purity
>99.99%
Bioactivity
MSC-4106, an orally active and potent YAP/TAZ-TEAD inhibitor, disrupts TEAD1 and TEAD3 auto-palmitoylation and demonstrates significant efficacy in the NCI-H226 tumor xenograft model [1].
Smiles
Cn1cc2c3cc(ccc3n(-c3ccc(cc3)C(F)(F)F)c2n1)C(O)=O
Molecular Formula
C18H12F3N3O2
Molecular Weight
359.3
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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