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Senexin A

Product Specifications

CAS Number

1366002-50-7

Target

CDK

Related Pathways

Cell Cycle/Checkpoint

Purity

0.9974

Bioactivity

Senexin A is an effective and selective CDK8 inhibitor that also inhibits CDK19 with Kd values of 0.83 microns and 0.31 microns, respectively.

Smiles

N#Cc1ccc2ncnc(NCCc3ccccc3)c2c1

Molecular Formula

C17H14N4

Molecular Weight

274.32

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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